Loading ...
with good selectivity over the 5-HT transporter(passive) have been discoveredhttp://dx.doi.org/10.1021/jm8001444 5-HT1 receptor antagonists
Nisijima , K. ; Yoshino , T. ; Yui , K. ; Katoh , S. Potent serotoninprevent5-ht)(2a ) receptor antagonists
Related Articles , Links Potent serotoninprevent5-HT)(2A ) receptor antagonists
through mutations within zalpha11 Ligand helix D.(passive) may be designedZalpha11 receptor antagonists
of three isoforms , one secreted ( sIL-1Rα / IL-1Rα1 ) , two intracellular ( IL-1Rα2 / IL-1Rα3 ) and produced by monocytes , tissue macrophages , Langerhans cells , dendritic cells , T and B cells , natural killer ( NK ) cells , large granular lymphocytes ( LGL ) , vascular endothelium , smooth muscle , fibroblasts , thymic epithelia , astrocytes , microglia , glioma cells , keratinocytes , and chondrocytes(passive) is composedreceptor antagonist ( IL-1RA
systolic(passive) is caused byaldosterone receptor antagonists
other branches(passive) might be caused byOrphenadrine , an NMDA receptor antagonist
for the management of insomnia(passive) have recently been discoveredOrexin - receptors antagonists
the endogenous agonist ( CXCL12(passive) preventing binding to the receptor and subsequent activation byReceptor antagonists
as a highly water - soluble agent keeping the selectivity and potency for AMPA receptors(passive) was discoveredAMPA receptor antagonist YM872
of three isoforms , one secreted ( sIL-1Ralpha / IL-1Ralpha1 ) , two intracellular ( IL-1Ralpha2 / IL-1Ralpha3(passive) is composedInterleukin-1 receptor antagonist ( IL-1RA
Oishi , Y , Nishimura , Y , Tanoue , Y , Kajihara , N , Imasaka , KI , Morita , S & Yasui , H 2005preventsEndothelin-1 receptor antagonist
AT1 andpreventedAT2 receptors antagonists
Blockade of these signaling pathways by CRF receptor antagonists ( Shaham et al . , 1998 ) orresultedhcrt receptor antagonists
some of which have recently entered clinical development(passive) have been discoveredPotent CXCR2 receptor antagonists
= naive mice lackingpreventsIL-1R. Interleukin-1 receptor antagonist ( IL-1Ra
to block the production of glutamate(passive) are designedThe NMDA receptor antagonists
PGD2(passive) caused byCRTH2 receptor antagonist
to block the excess endothelin by various means(passive) are designedEndothelin receptor antagonists
Merck &(passive) originated byCGRP ) receptor antagonist
2014;289:10399 - 410 pubmed publisher Davidowa H , Ziska TpreventPlagemann A. GABAA receptor antagonists
Statistical comparisons of effects of ionotropic receptor blockade Across the sample of neuronscontributedmajor ionotropic receptor antagonists
to interfere with the interaction between HIV-1 and its co - receptors(passive) have been designedCo - receptor antagonists
to promote aquaresis(passive) are designedreceptor antagonists
to become novel important pharmacological tools within the current therapeutic repertoire available for the management of various inflammatory conditions(passive) are setChemokine receptor antagonists
some measuresto leadto a histamine-1 receptor antagonists
a marketleading5-HT3 receptor antagonist
based on tyrosine derivatives(passive) are being designedAntagonists of the P2X7 receptor
either video sekseiinfluenceadrenergic receptor antagonists
Removal of extracellular magnesium or addition oftriggeredGABA receptor antagonists
to block vasoconstricting peptides , which are believed to play an important role in essential hypertension(passive) are designedEndothelin receptor antagonists
to lower plasma glucose levels(passive) are designedGlucagon receptor antagonists
Briyal , S. , Philip , T. and GulatipreventA. Endothelin - A receptor antagonists
Schering - Plough(passive) discovered byA₂A receptor antagonist
This hypothetic mechanism of action of gastrin resulted in a strategyto rationally designgastrin receptor antagonists
to lower glucose levels by reducing the production of glucose by the liver(passive) are designedGlucagon receptor antagonists
Belanger MC , ( 1998influenceNMDA receptor antagonists
Local application of specific NMDA , AMPA , orresultsGABAA receptor antagonists
Adenosine Therapeutics(passive) discovered byAdenosine Receptor Antagonists
combining responses to soft and loud stimulimay leadto NMDA receptor antagonists
completelypreventcompletely
the induction of interneuron LTDalso preventedthe induction of interneuron LTD
neuronal death in cell culture(passive) can be prevented byneuronal death in cell culture
NSAID - induced exacerbations in patients with chronic urticariamay preventNSAID - induced exacerbations in patients with chronic urticaria
anos effect of capsaicinpreventanos effect of capsaicin
intracellular Ca2 + overload and neuronal death(passive) can be prevented byintracellular Ca2 + overload and neuronal death
amyloid - β - induced increase in ETA receptor expression , oxidative stress , and cognitive impairmentpreventamyloid - β - induced increase in ETA receptor expression , oxidative stress , and cognitive impairment
acute inflammation in vivo ... 33preventacute inflammation in vivo ... 33
sudden death in heart failureto preventsudden death in heart failure
the development of pulmonary emphysema in rats Y Chen · M Hanaokapreventthe development of pulmonary emphysema in rats Y Chen · M Hanaoka
Both receptor internalization and down - regulation(passive) were prevented byBoth receptor internalization and down - regulation
the effects of acetylcholinepreventthe effects of acetylcholine
the opposite effectscausedthe opposite effects
the anticonvulsant effects of ( +preventedthe anticonvulsant effects of ( +
unexpected effectsmay causeunexpected effects
Expert review of liver injury(passive) caused byExpert review of liver injury
the neuronal death associated with repeated brief ischemia ... Kato et al . ... 1990preventthe neuronal death associated with repeated brief ischemia ... Kato et al . ... 1990
cisplatin - induced emesis in Cryptotis parva ... a new experimental model of emesispreventcisplatin - induced emesis in Cryptotis parva ... a new experimental model of emesis
both normal developmental neuronal death and deafferentation - induced death in the auditory nuclei of chick embryospreventboth normal developmental neuronal death and deafferentation - induced death in the auditory nuclei of chick embryos
the development of pulmonary emphysema in rats ... ” European Respiratory Journal , volpreventthe development of pulmonary emphysema in rats ... ” European Respiratory Journal , vol
not only the vascular tone , but also the inappropriate VSMC growth , which occurs in pathological cardiovascular conditionsmay influencenot only the vascular tone , but also the inappropriate VSMC growth , which occurs in pathological cardiovascular conditions
neuronal death.10 Administration of perampanel results in rapid and complete absorption with negligible first - pass metabolismmay preventneuronal death.10 Administration of perampanel results in rapid and complete absorption with negligible first - pass metabolism
both acute and delayed chemotherapy - induced nausea and vomitingpreventboth acute and delayed chemotherapy - induced nausea and vomiting
beta - amyloid ( 25 - 35)-induced cognitive deficits in mice memory | A(2A ) receptor | ALZHEIMERS - DISEASE | INVOLVEMENT | RELEASE | NEUROTOXICITY | NEUROSCIENCES | NUCLEUS - ACCUMBENS | adenosine | beta - amyloid | HIPPOCAMPUS | caffeine | neuroprotection | GLUTAMATE |preventbeta - amyloid ( 25 - 35)-induced cognitive deficits in mice memory | A(2A ) receptor | ALZHEIMERS - DISEASE | INVOLVEMENT | RELEASE | NEUROTOXICITY | NEUROSCIENCES | NUCLEUS - ACCUMBENS | adenosine | beta - amyloid | HIPPOCAMPUS | caffeine | neuroprotection | GLUTAMATE |
acute respiratory distress syndrome and death ... implications for Coronavirus disease 2019preventacute respiratory distress syndrome and death ... implications for Coronavirus disease 2019
The yawning evoked by an a - MSH - related peptide , ACTH , which was unaffected by oxytocin receptor antagonists , was also reported(passive) to be prevented byThe yawning evoked by an a - MSH - related peptide , ACTH , which was unaffected by oxytocin receptor antagonists , was also reported
the toxic effect of these ADDLsmight preventthe toxic effect of these ADDLs
central sensitization induced by peripheral nociceptive stimulation and abolish hypersensitization once it is established9 by blocking dorsal horn NMDA receptor activation induced by excitatory amino acid transmitters , such as glutamate and aspartate9 - 11preventcentral sensitization induced by peripheral nociceptive stimulation and abolish hypersensitization once it is established9 by blocking dorsal horn NMDA receptor activation induced by excitatory amino acid transmitters , such as glutamate and aspartate9 - 11
parathyroid cell proliferation caused by hypocalcemia in ratspreventparathyroid cell proliferation caused by hypocalcemia in rats
blood vessels from narrowing Phosphodiesterase Inhibitors ( PDE 5 Inhibitorspreventblood vessels from narrowing Phosphodiesterase Inhibitors ( PDE 5 Inhibitors
the development of the tolerance to analgesic effects of kappa opioids ( Bhargava and Thorat , 1994;Bhargava et al . , 1995preventthe development of the tolerance to analgesic effects of kappa opioids ( Bhargava and Thorat , 1994;Bhargava et al . , 1995
atorvastatin antidepressant - like effectpreventedatorvastatin antidepressant - like effect
emesis associated with serotonin release from the gastrointestinal tract occurring in gastroenteritis ( Cubeddu et al .preventemesis associated with serotonin release from the gastrointestinal tract occurring in gastroenteritis ( Cubeddu et al .
some of the acute behavioral effects of 3,4-methylenedioxymethamphetaminecould preventsome of the acute behavioral effects of 3,4-methylenedioxymethamphetamine
the development of pulmonary emphysema in rats First Dept of Medicine , Shinshu University School of Medicine , Asahi , Matsumoto , Japan Eur Respir J 35:904 - 12preventthe development of pulmonary emphysema in rats First Dept of Medicine , Shinshu University School of Medicine , Asahi , Matsumoto , Japan Eur Respir J 35:904 - 12
pathological damage to astrocytes,[60preventpathological damage to astrocytes,[60
This effect of airway jugular C - fiber activation(passive) was prevented byThis effect of airway jugular C - fiber activation
aerosol agonist - induced bronchospasm and antigen - evoked airways hyperresponsiveness ( effects(passive) are prevented byaerosol agonist - induced bronchospasm and antigen - evoked airways hyperresponsiveness ( effects
this sensitizing effect of nociceptor stimulation.110Similar sensitizing effects of nociceptor stimulation on cough may be evoked from the esophagus , and observation that may explain how GERD initiatespreventthis sensitizing effect of nociceptor stimulation.110Similar sensitizing effects of nociceptor stimulation on cough may be evoked from the esophagus , and observation that may explain how GERD initiates
the anticonvulsive effects mediated by Ang IV or LVV - H7 , the recovery of the sst2A receptors at the plasma membranepreventthe anticonvulsive effects mediated by Ang IV or LVV - H7 , the recovery of the sst2A receptors at the plasma membrane